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. Author manuscript; available in PMC: 2016 Mar 27.
Published in final edited form as: Angew Chem Int Ed Engl. 2015 Feb 9;54(14):4226–4230. doi: 10.1002/anie.201411901

Scheme 1.

Scheme 1

General scheme for RebH catalyzed halogenation and substrates used for directed evolution via substrate walking.