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. 2015 Jun 11;12(8):2912–2923. doi: 10.1021/acs.molpharmaceut.5b00173

Table 2. IC50 Values of Various Formulations of Tvlocrebrine in A431 and A549 Cells.

A431 cells IC50 at physiological pH (nM) IC50 at acidic pH (nM)
free drug 210 432
nontargeted nanoparticles 154 132
targeted nanoparticles 31 28
A549 cells IC50 at physiological pH (nM) IC50 at acidic pH (nM)
free drug 37 361
nontargeted nanoparticles 28 47
targeted nanoparticles 7 24