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Fluorescence polarization assay binding data (Ki values in μM)
| ||
|---|---|---|
| inhibitor | R | Ki (μM) |
| 7 |
|
15.5 ± 4.7 |
| 17b |
|
8.0 ± 2.4 |
| 17c |
|
6.2 ± 2.0 |
| 17e |
|
26.5 ± 0.4 |
| 17f |
|
41.0 ± 0.4 |
| 17g |
|
13.3 ± 0.6 |
| 17h |
|
> 100 |
| 17i |
|
30.6 ± 11 |
| 17k |
|
11.0 ± 0.3 |
| 17o |
|
12.8 ± 0.3 |
