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. Author manuscript; available in PMC: 2016 Jan 31.
Published in final edited form as: Bioorg Med Chem Lett. 2014 Dec 13;25(3):690–694. doi: 10.1016/j.bmcl.2014.11.082

Table 3.

Structures and activities of matrix library analogs 7.

graphic file with name nihms649279t27.jpg Ar1
Entry hM5IC50
(µM)a 		hM5IC50
(µM)a 		hM5IC50
(µM)a
1 3.2 >30 4.1 graphic file with name nihms649279t28.jpg
2 >30 2.4 1.9 graphic file with name nihms649279t29.jpg
3 1.3 1.0 1.1 graphic file with name nihms649279t30.jpg
4 3.3 >30 3.2 graphic file with name nihms649279t31.jpg
5 5.5 1.4 3.3 graphic file with name nihms649279t32.jpg
6 1.2 0.51 1.3 graphic file with name nihms649279t33.jpg
7 2.7 0.7 1.3 graphic file with name nihms649279t34.jpg
8 2.0 1.6 6.4 graphic file with name nihms649279t35.jpg
9 1.3 0.9 2.2 graphic file with name nihms649279t36.jpg
a

hM5 IC50 data, n = 1; hM5 IC50 for 7B-6, n = 6, pIC50 = 6.29±0.02