Table 1.
compound | % inhibition in screen | CC50 (μM) | IC50 (μM) | SI (CC50/IC50) | |
---|---|---|---|---|---|
1 | lanatoside C | 100.0 | 0.177 | 0.255 | 0.694 |
2 | gambogic amide | 100.0 | 0.454 | 1.01 | 0.45 |
3 | strophanthidin | 100.0 | 0.491 | 1.161 | 0.423 |
4 | acetyl isogambogic acid | 99.0 | 2.885 | 2.935 | 0.983 |
5 | puromycin hydrochloride | 99.7 | 3.594 | 0.889 | 4.043 |
6 | emetine | 98.3 | >50 | 1.474 | >33.921 |
7 | plumbagin | 98.3 | 0.756 | 0.919 | 0.823 |
8 | cycloheximide | 97.9 | >50 | 0.608 | >82.237 |
9 | digitoxin | 92.5 | 0.031 | 0.05 | 0.62 |
10 | crinamine | 91.5 | >50 | 3.789 | >13.196 |
11 | mycophenolic acid | 90.5 | >50 | 0.316 | >158.228 |
12 | cantharidin | 87.3 | >50 | 11.325 | >4.415 |
13 | azacitidine | 76.9 | >50 | 4.011 | >12.466 |
14 | gedunin | 72.9 | 5.484 | 0.803 | 6.829 |
15 | fluorouracil | 70.6 | >50 | >50 | |
16 | methotrexate | 67.1 | >50 | >50 | |
17 | gemfobrozil | 62.1 | >50 | >50 | |
18 | dramamine | 57.8 | >50 | >50 | |
19 | vidarabine | 56.1 | >50 | >50 |