Table 1. Activity of the 15 Test Compounds in the Plasmid-Based Enzymatic Assay with PA-Nter.
compd | IC50 (μM)a | compd | IC50 (μM)a |
---|---|---|---|
1 | >500 | 9 | >500 |
2 | >500 | 10 | 0.94 |
3 | >500 | 11 | 65 |
4 | >500 | 12 | >500 |
5 | >500 | 13 | >500 |
6 | >500 | 14 | >500 |
7 | >500 | 15 | 7.0 |
8 | >500 | L-742,001 | 0.48 |
IC50: 50% inhibitory concentration, calculated using nonlinear regression analysis. Values are the result of at least three independent experiments.