Table 4. Selectivity Data for Compound 1j.
| IC50 (μM) | fold of selectivity | |
|---|---|---|
| ADAMTS-4 | 0.01 | |
| ADAMTS-5 | >10 | >1000 |
| ADAMTS-13 | >10 | >1000 |
| MMP-13 | >10 | >1000 |
| TACE | >10 | >1000 |
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