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| metabolic stability (T1/2 min) | 49 (H), 108 (M), 69 (R), 70 (D) |
| PAMPA (pH 7.4) | 698 nm/sec |
| HLM CYP IC50 | all >40 μM; except CYP3A4 (3 μM) and 1A2 (1 μM) |
| hERG patch clamp | 20% inh at 30 μM |
| Na+ patch clamp | <10% inh at 10 μM (1 Hz and 4 Hz) |
| Ca2+ patch clamp IC50 | >80 μM |
| PXR EC50 | >50 μM |
| HEPG2 IC50 | >50 μM |
