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. 2015 Jul 12;6(8):850–855. doi: 10.1021/acsmedchemlett.5b00226

Table 4. Pharmacokinetic Profile of BMS-911543.

PK mousea ratb dogc cynod
CL (mL/min/kg) 0.55 0.7 6.5 5.3
Vss (L/kg) 0.26 0.3 1.6 1.1
T1/2 (h) 5.1 5 2.2 2.4
F (%) 100 100 82 53
a

Mice were dosed 2.0 mg/kg IV and 10.0 mg/kg PO.

b

Rats were dosed 1.0 mg/kg IV and 1.0 mg/kg PO.

c

Dogs were dosed 0.2 mg/kg IV and 0.2 mg/kg PO.

d

Cyno were dosed 1.0 mg/kg IV and 1.0 mg/kg PO.