Table 3.
Compound | HT-29c | NF-κB (p65)d | P. falciparume |
---|---|---|---|
1 | > 20 | > 20 | 0.65 ± 0.06 |
2 | 13.2 | > 20 | 1.28 ± 0.13 |
3 | 3.3 | > 20 | 1.02 ± 0.09 |
4 | > 20 | > 20 | 0.26 ± 0.01 |
5 | 18.4 | > 20 | 0.63 ± 0.02 |
6 | > 20 | > 20 | > 10 |
7 | 1.9 | > 20 | 2.07 ± 0.13 |
8 | > 20 | > 20 | > 10 |
9 | > 20 | 4.0 | 1.33 ± 0.37 |
Paclitaxelf | 0.001 | - | - |
Rocaglamideg | - | 0.08 | - |
Artemisininh | - | - | 0.0007 |
No obvious growth inhibition of C. albicans cells were observed for the test compounds at a concentration of 40 mg/mL.
Results are expressed as ED50 or IC50 values (µM).
Compounds with ED50 values of > 20 µM in HT-29 cells are considered inactive.
Compounds with IC50 values of > 20 µM on an enzyme-based ELISA NF-κB (p65) assay are considered inactive.
Compounds with IC50 values of > 10 µM in P. falciparum assay are considered inactive.
Used as a positive control substance for the cytotoxicity assay.
Used as a positive control substance for the cytotoxicity assay.
Used as a positive control substance for the P. falciparum assay.