Table 2.
Scope of the tandem CEYM-IMDAR protocol.
![]() | |||
| entry | 1 (R) | 2 | 3 (yield)a |
| 1 | 1a (H) |
![]() 2a |
![]() 3a (57%) |
| 2 | 1a (H) |
![]() 2b |
![]() 3b (38%) |
| 3 | 1a (H) |
![]() 2c |
![]() 3c (62%) |
| 4 | 1b (F) |
![]() 2c |
![]() 3d (45%) |
| 5 | 1c (OMe) |
![]() 2c |
![]() 3e (35%) |
| 6 | 1a (H) |
![]() 2d |
![]() 3f (50%) |
| 7 | 1a (H) |
![]() 2e |
![]() 3g (44%) |
aIsolated yields after column chromatography. All final products 3 were obtained as single diastereoisomers.














