Table 4.
Doses of MP-10 (mg/kg) | Kinetic parameters (Striatum) | |||||
---|---|---|---|---|---|---|
LoganREF | SRTM | |||||
BPND | Occ% | BPND | R1 | k2 (min−1) | Occ % | |
2.00 | 0.4231 | 89.23 | 0.6558 | 1.0209 | 0.04245 | 86.65 |
1.50 | 0.4234 | 89.17 | 0.5732 | 0.8844 | 0.08179 | 80.00 |
1.00 | 0.8980 | 77.14 | 0.9026 | 0.9932 | 0.05868 | 81.63 |
0.50 | 0.8214 | 79.09 | 1.3084 | 0.7716 | 0.08542 | 73.37 |
0.25 | 2.8957 | 26.26 | 3.8161 | 1.0628 | 0.08540 | 22.32 |
0.10 | 3.7678 | 4.06 | 4.0338 | 1.1128 | 0.10847 | 17.79 |
0.05 | 3.7307 | 5.01 | 4.0253 | 0.9354 | 0.09479 | 18.07 |