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. 2015 Oct 16;7(10):4175–4198. doi: 10.3390/toxins7104175
Compd. No. R1 R2 Radioligand Displacement Assay IC50 (μM) SH-SY5Y Neuroblastoma Cells IC50 (μM) HEK293 hCav2.2 + β3 + α2δ1 IC50 (μM)
25 H NH2 214 160 232
26 H N=C(NH2)2 12 206 299
27 F NH2 65 286 288
28 F N=C(NH2)2 16 156 156