Table 1. Characterization of IMPDHs from filamentous fungi.
IC50 (MPA) (μM) | kcat (s−1) | KM (IMP) (μM) | kcat/KM (IMP) (M−1s−1) | KM (NAD+) (μM) | kcat/KM (NAD) (M−1s−1) | Kü (NAD+) (mM) | |
---|---|---|---|---|---|---|---|
AnImdA | 0.026 ± 0.002 | 0.74 ± 0.06 | 10 ± 1 | 74,000 ± 8,000 | 170 ± 70 | 4,400 ± 100 | 1.5 ± 0.6 |
PbIMPDH-A | 0.43 ± 0.03 | 0.70 ± 0.08 | 130 ± 30 | 5,400 ± 1,200 | 340 ± 90 | 2,100 ± 900 | 4.7 ± 1.1 |
PbIMPDH-B | 27 ± 9 | 0.41 ± 0.02 | 1,400 ± 200 | 300 ± 80 | 790 ± 140 | 500 ± 100 | n.a. |
PcIMPDH-A | 0.036 ± 0.004 | 0.84 ± 0.03 | 40 ± 6 | 21,000 ± 2,000 | 290 ± 60 | 2900 ± 300 | 2.4 ± 0.5 |
PcIMPDH-B | 0.06 ± 0.01 | 0.0075 ± 0.001 | 600 ± 300 | 12 ± 3 | 640 ± 130 | 11 ± 6 | n.a. |