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. 2015 Nov 14;593(22):4943–4961. doi: 10.1113/JP270971

Table 2.

The inhibition site is not enantioselective

XmTFD‐MPPB k –1 (s–1) k +1 (×105 m −1 s–1) K Dm) Recovery (s−1)
S,10 μmGABA 2.0 ± 0.32 1.0 ± 0.12∗∗ 20 ± 4.0 2 ± 0.2
S,10 mmGABA 2.1 ± 0.24 0.43 ± 0.08 52 ± 11 6.9 ± 0.5
R,10 mmGABA 1.6 ± 0.38 0.34 ± 0.1 48 ± 20

Data are shown as mean ± SD.

*k –1 values do not differ.

**k +1 at 10 μm and 10 mm are different (P < 0.001).