Table 2.
Affinity of PWZ-029 (1); K i (nM)a.
| Code | MW | α1 | α2 | α3 | α4 | α5 | α6 |
|---|---|---|---|---|---|---|---|
| PWZ-029 (1) | 291.73 | >300 | >300 | >300 | ND | 38.8 | >300 |
| PWZ-029 (1) | 291.73 | 920 | ND | ND | ND | 30 | ND |
| PWZ-029 (1) | 291.73 | 362 | 180 | 328 | ND | 6 | ND |
aData from three separate laboratories.
Affinity of PWZ-029 (1); K i (nM)a.
| Code | MW | α1 | α2 | α3 | α4 | α5 | α6 |
|---|---|---|---|---|---|---|---|
| PWZ-029 (1) | 291.73 | >300 | >300 | >300 | ND | 38.8 | >300 |
| PWZ-029 (1) | 291.73 | 920 | ND | ND | ND | 30 | ND |
| PWZ-029 (1) | 291.73 | 362 | 180 | 328 | ND | 6 | ND |
aData from three separate laboratories.