Skip to main content
. 2015 Nov 12;137(47):14861–14864. doi: 10.1021/jacs.5b10221

Table 2. Scope of Dearomative Indole (3 + 2) Reactiona.

graphic file with name ja-2015-10221v_0010.jpg

graphic file with name ja-2015-10221v_0011.jpg

a

Indole (1 equiv), α-haloamide (2 equiv), Na2CO3 (4 equiv) in HFIP, 0.25 M.

b

Isolated yield.

c

Significant decomposition products observed.