Table 1. Inhibitor constant (Ki) values in Molar (M) range of EgKI-1 and EgKI-2.
Inhibitor | Trypsin | Chymotrypsin | Pancreatic elastase | Neutrophil elastase | Cathepsin G | |||||
---|---|---|---|---|---|---|---|---|---|---|
Ki (M) | CI95 | Ki (M) | CI95 | Ki (M) | CI95 | Ki (M) | CI95 | Ki (M) | CI95 | |
EgKI-1 | 2.32x10-7 | 0.17–0.28 | 1.484x10-9 | 0.20–0.62 | 1.65x10-9 | 1.23–2.06 | 6.42x10-11 | 32.74–95.66 | 4.47x10-10 | 0.20–0.62 |
EgKI-2 | 1.38x10-8 | 9.84–17.8 | NI | NI | NI | NI | NI | NI | NI | NI |
NI- No inhibition,
CI95- 95% confidence interval.