Table 1. Specificity of 9 for mPTPB over a Panel of PTPs.
PTP | IC50 |
---|---|
mPTPB | 18 ± 2 nM |
mPTPA, PTP1B, TC-PTP, LYP, HePTP, SHP1, SHP2, PTPH1, Meg2, FAP1, CD45, LAR, PTPα, PTPβ, PTPγ, PTPμ, PTPε, PTPσ, MKP5, VHR, VHX, CDC14A, Laforin, LMWPTP, PP5 | no inhibition at 200 μM |