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. 2015 Nov 3;6(12):1231–1235. doi: 10.1021/acsmedchemlett.5b00373

Table 1. Specificity of 9 for mPTPB over a Panel of PTPs.

PTP IC50
mPTPB 18 ± 2 nM
mPTPA, PTP1B, TC-PTP, LYP, HePTP, SHP1, SHP2, PTPH1, Meg2, FAP1, CD45, LAR, PTPα, PTPβ, PTPγ, PTPμ, PTPε, PTPσ, MKP5, VHR, VHX, CDC14A, Laforin, LMWPTP, PP5 no inhibition at 200 μM