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. 2015 Dec 31;60(1):229–238. doi: 10.1128/AAC.02157-15

TABLE 7.

Activity of azoles in C. albicans multidrug transporter mutants

C. albicans transporter mutant Resistance mechanism/genotype MIC (μg/ml)
Fluconazole Itraconazole Posaconazole Voriconazole Isavuconazole
CAF2-1 URA3/ura3Δ 0.25 0.0625 0.0625 <0.0039 0.0078
DSY448 cdr1Δ/Δ <0.0625 0.0625 0.0625 <0.0039 <0.001
DSY465 mdr1Δ/Δ 0.25 0.0625 0.0625 <0.0039 0.0078
DSY468 cdr1Δ/Δ mdr1Δ/Δ <0.0625 0.0625 0.0156 <0.0039 <0.001
DSY653 cdr2Δ/Δ 0.125 0.0625 0.0156 <0.0039 0.0078
DSY654 cdr1Δ/Δ cdr2Δ/Δ <0.0625 0.0156 0.0156 <0.0039 0.002
DSY1054 flu1Δ/Δ 0.25 0.0625 0.0625 <0.0039 0.0156
DSY1021 cdr1Δ/Δ cdr2Δ/Δ flu1Δ/Δ <0.0625 0.0625 0.0625 <0.0039 <0.001
DSY1024 cdr1Δ/Δ cdr2Δ/Δ flu1Δ/Δ mdr1Δ/Δ <0.0625 0.0156 0.125 <0.0039 <0.001
DSY1050 cdr1Δ/Δ cdr2Δ/Δ mdr1Δ/Δ <0.0625 0.0156 0.0312 <0.0039 0.002
DSY1055 flu1Δ/Δ mdr1Δ/Δ 0.25 0.0156 0.125 <0.0039 0.0156