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| Probe | Target | Mode of action |
|---|---|---|
| (+)-JQ1, I-BET, PFI-1 (ref. 4) | BET family bromodomains | Inhibitor |
| Rapamycin | mTOR | Allosteric inhibitor |
| GW683965 (ref. 12) | LXRα and LXRβ | Agonist |
| PF-04457845 (ref. 34) | Fatty acid amide hydrolase | Irreversible inhibitor |
| GNF-5 (ref. 35) | Bcr-Abl | Allosteric inhibitor |
| Cyclopamine | Smoothened | Orthosteric inhibitor |
