Table 5.
BACE1 Inhibition
Comp. | Name | μM | % Inhibition |
---|---|---|---|
1 | Purpuramine M | 42.0 | 36 |
3 | Araplysillin VII | 39.6 | 40 |
5 | Araplysillin IX | 41.9 | 35 |
6 | Araplysillin X | 31.4 | 70 |
7 | Araplysillin XI | 30.6 | 60 |
8 | Hexadellin A | 41.7 | 27 |
9 | Araplysillin II | 31.8 | 57 |
11 | Purpurealidin I | 42.0 | 74 |
12 | Aplysamine 4 | 42.6 | 62 |
13 | Purpuramine G | 48.3 | 48 |
Secretase Inhibitor IV | 0.021 | 80 |