Table 1. Effects of C4 Modification on Potency and wtEGFR Selectivity.
Ki data are an average of at least two independent experiments.
Ratio of wtEGFR Kiapp over EGFR(TMLR) Kiapp.
Ki data are an average of at least two independent experiments.
Ratio of wtEGFR Kiapp over EGFR(TMLR) Kiapp.