| Nomenclature | NTS1 receptor | NTS2 receptor |
| HGNC, UniProt | NTSR1, P30989 | NTSR2, O95665 |
| Rank order of potency | neurotensin (NTS, P30990) >neuromedin N {Mouse, Rat} [741] | neurotensin (NTS, P30990) = neuromedin N {Mouse, Rat} [1235] |
| Selective agonists | JMV449 (pK i 10) [1753] – Rat | levocabastine (pK i 6.8) [1235, 1583] |
| Antagonists | meclinertant (pIC50 7.5–8.2) [664] | – |
| Labelled ligands | [3H]meclinertant (Antagonist) (pK d 8.5) [1030] – Rat | – |
| Comments | – | A splice variant of the NTS2 receptor bearing 5 transmembrane domains has been identified in mouse [191] and later in rat [1492]. |
Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.