Nomenclature	kisspeptin receptor
HGNC, UniProt	KISS1R, Q969F8
Endogenous agonists	kisspeptin‐10 (KISS1) (Selective) (pK i 8.6–10.4) [996, 1434], kisspeptin‐54 (KISS1, Q15726) (Selective) (pK i 8.8–9.5) [996, 1434], kisspeptin‐14 (KISS1, Q15726) (pK i 8.8) [996], kisspeptin‐13 (KISS1, Q15726) (Selective) (pK i 8.4) [996]
Selective agonists	4‐fluorobenzoyl‐FGLRW‐NH2 (pEC50 9.2) [1894], [dY]1KP‐10 (pIC50 8.4) [385] – Mouse
Selective antagonists	peptide 234 [1600]
Labelled ligands	[125I]Tyr45‐kisspeptin‐15 (Agonist) (pK d 10) [1434], [125I]kisspeptin‐13 (human) (Agonist) (pK d 9.7) [1252], [125I]kisspeptin‐10 (human) (Agonist) (pK d 8.7) [996], [125I]kisspeptin‐14 (human) (Agonist) [1252]