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. 2016 Jan 7;22(5):1614–1617. doi: 10.1002/chem.201504636

Table 2.

Substrate scope of the iodine(III)-mediated thioamination.

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Entry Substrate Nucleophile Product Yield [%]
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1 1 a (R=H) PhSNa 2 a (R=H) 79
2 3 (R=Cl) PhSNa 4 (R=Cl) 75
3 5 (R=OMe) PhSNa 6 (R=OMe) 70
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4 7 PhSNa 8 60
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5 9 PhSNa 10 71
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6 11 PhSNa 12 56
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7 11 Inline graphic 13 57
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8 11 Inline graphic 14 50