Table 2.
Entry | Substrate | Nucleophile | Product | Yield [%] |
---|---|---|---|---|
1 | 1 a (R=H) | PhSNa | 2 a (R=H) | 79 |
2 | 3 (R=Cl) | PhSNa | 4 (R=Cl) | 75 |
3 | 5 (R=OMe) | PhSNa | 6 (R=OMe) | 70 |
4 | 7 | PhSNa | 8 | 60 |
5 | 9 | PhSNa | 10 | 71 |
6 | 11 | PhSNa | 12 | 56 |
7 | 11 | 13 | 57 | |
8 | 11 | 14 | 50 |