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. Author manuscript; available in PMC: 2016 Nov 15.
Published in final edited form as: Bioorg Med Chem. 2015 Nov 15;23(22):7226–7233. doi: 10.1016/j.bmc.2015.10.019

Fig. 5.

Fig. 5

Proposed mechanism and functional outcome of inhibition of NPM1 by the 1-benzyl-2-methyl-3-indolylmethylene barbituric acid analogue YTR-107 (1) and 1-benzyl-2-methyl-3-indolylmethylene thio barbituric acid analogue PNR-605 (7l).