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. 2016 Jan 29;60(2):797–805. doi: 10.1128/AAC.00426-15

FIG 1.

FIG 1

General synthesis of N-acylated trans-aziridine-2,3-dicarboxylates. Reagents and conditions are as follows: i, PPA, ethyl acetate, or dimethylformamide, 1 h at 0°C and 24 h at room temperature (s1 to s37); and ii, PPA, triethylamine, or ethyl acetate, 1 h at 0°C, 4 h at 40°C, and 7 days at room temperature (s38).