Table 1.
Cell Line | CFZ IC50 (nM) | SAHA IC50 (nM) | CFZ+SAHA IC50 (nM) | Combination Index | ||||
---|---|---|---|---|---|---|---|---|
48 h | 72 h | 48 h | 72 h | 48 h | 72 h | 48 h | 72 h | |
H520 | 15.13 | 1.10 | 20251 | 8941 | 8.13 | 0.59 | 0.30 | 0.26 |
A549 | 127.3 | 104.8 | 6871 | 6340 | 11.38 | 17.89 | 0.19 | 0.29 |
H1993 | 12.94 | 5.36 | 8103 | 6827 | 6.66 | 4.40 | 0.35 | 0.68 |
H460 | 56.50 | 41.21 | 10448 | 7203 | 22.06 | 20.82 | 0.21 | 0.33 |
H1299 | 8.03 | 16.30 | 25609 | 24418 | 10.52 | 11.46 | 0.87 | 0.76 |
The determined inhibitory concentrations (IC50 values) represent the level of drug that inhibited cell growth by 50%. IC50 values (nM) are the mean of one experiment, n=6. Combination index (CI) values were obtained by the method described by Chou and Talalay (1983). Values shown are an average CI from a single experiment at growth inhibition rates of 50%, 75%, 90% and 95%. CI interpretation: <0.3 = strong synergism, 0.3-0.7 = synergism, 0.7-0.9 = moderate to slight synergism, 0.9-1.1 = nearly additive, 1.1-1.45 slight to moderate antagonism.