Table 1. Quantitative analysis of UNC3866 binding to CBX and CDY chromodomains by ITC.
Chromodomain | UNC3866 Kd (μM) |
---|---|
CBX2 | 1.8 ± 0.21 |
CBX4 | 0.094 ± 0.017 |
CBX6 | 0.610 ± 0.0078 |
CBX7 | 0.097 ± 0.0024 |
CBX8 | 1.2 ± 0.021 |
CDY1 | 6.3 ± 0.92 |
CDYL1b | 0.91 ± 0.076 |
CDYL2 | 0.85 ± 0.076 |