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. Author manuscript; available in PMC: 2016 Feb 25.
Published in final edited form as: Drug Discov Today. 2006 Dec 20;12(0):132–138. doi: 10.1016/j.drudis.2006.12.011

Figure 3.

Figure 3

Schematic representation of simulated transitions between the three protease forms. The closed flap conformation converts to semi-open upon removal of ligand. Ligand induces the closure of the open form. Free protease exists primarily in semi-open form but transiently changes to fully open and, occasionally, even to the closed form that is only weakly populated in the absence of a ligand.