Table 2.
Population pharmacokinetic parameter values ± standard deviation estimated in dihydropyrimidine dehydrogenase (DPD)‐deficient subjects (EURDEF model), subjects with normal DPD activity (EURNOR model) and all subjects (EURMIX model)
Km (mg l −1 ) | V max (mg h −1 *1.85m −2 ) | ka po (h −1 ) | V(l) | |
---|---|---|---|---|
EURDEF | 5.99 ± 4.17 | 494 ± 133 | 5.61 ± 7.16 | 0.57 ± 0.09 |
EURNOR | 7.69 ± 1.38 | 837 ± 130 | 4.65 ± 3.33 | 0.51 ± 0.14 |
EURMIX | 7.10 ± 3.33 | 641 ± 178 | 5.13 ± 4.87 | 0.55 ± 0.12 |
Ka, absorption constant; Km, Michaelis–Menten constant; po, per oral; V, apparent volume of drug distribution; Vmax, maximum enzymatic conversion capacity.