Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
Selected Pyridinone Analogs Acting as GSK-3β Inhibitors
*The number written inside the parenthesis corresponds to the number/code given to the compounds in their original publication.
aGSK-3β cell-free enzyme inhibition assay.
bGSK-3β whole-cell enzyme inhibition assay.
cCNS multi-parameter optimization (MPO) score. A score >4.5 indicates an increased probability of CNS penetration.
