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. Author manuscript; available in PMC: 2016 Mar 7.
Published in final edited form as: Bioorg Med Chem. 2013 Jan 30;21(7):1787–1794. doi: 10.1016/j.bmc.2013.01.049

Figure 2. BrSAH is a potent inhibitor of DOT1L.

Figure 2

IC50 values for 5-ITC, SAH and BrSAH were determined (18.4, 0.6 and 0.077 μM respectively) at Km of SAM, using a radioactivity based assay as described in material and methods.