Table 2.
Compound Set | N [number] | NG [molecular graphs] | NG /N [diversity ratio] | Ns [singleton graphs] | Ns/N [singleton ratio] |
---|---|---|---|---|---|
NCI Diversity Set III | 1560 | 652 | 0.42 | 475 | 0.31 |
HTVS-SP-XP-NN2/Antagonist | 15 | 15 | 1.0 | 15 | 1.0 |
HTVS/Agonist | 15 | 14 | 0.93 | 13 | 0.87 |
HTVS-SP-XP-NN1/Agonist | 15 | 13 | 0.87 | 12 | 0.80 |
N = total number of compounds in the library, NG = number of molecular graphs in the library, NG/N = diversity ratio, Ns = number of singleton molecular graph scaffolds, Ns/N = singleton ratio.