Table 4.
Dose level
|
|||||
---|---|---|---|---|---|
1A | 1 | 2 | 3 | 4 | |
No. of patients | 3 | 3 | 6 | 6 | 3 |
Oxaliplatin | 60 mg/m2 | 60 mg/m2 | 60 mg/m2 | 60 mg/m2 | 60 mg/m2 |
Irinotecan | 40 mg/m2 | 40 mg/m2 | 40 mg/m2 | 50 mg/m2 | 60 mg/m2 |
Capecitabine | 1,000 mg bid | 300 mg bid | 450 mg bid | 450 mg bid | 450 mg bid |
Free platinum Cmax Mean (SD, CV %) | 0.85 (0.15,18) | 0.65 (0.15, 23) | 0.72 (0.16, 22) | 0.76 (0.19, 25) | 1.34 (0.42, 31) |
Free Platinum AUC Mean (SD, CV %) | 8.5 (2.2, 26) | 11.0 (10.3, 94) | 9.2 (10.8, 117) | 3.4 (2.4, 71) | 7.3 (3.2, 44) |
Free Platinum Cl (mL/min) Mean (SD, CV %) | 120.3 (41.1, 34) | 144.2 (89.8, 62) | 198.1 (118.4, 60) | 294.5 (116.3,40) | 142.2 (97.0, 68) |