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. 2016 Feb 24;8(1):5. doi: 10.3390/pharmaceutics8010005

Figure 1.

Figure 1

Inhibition of CYPs. Concentration-dependent effect of venetoclax (0.01–20 µM) on the enzyme activity of CYP2B6, CYP2C19, and CYP3A4. Data are expressed as mean ± SEM for n = 3 biological replicates measured in duplicate. CYPs with no inhibition (CYP1A2, CYP2D6) are not depicted.