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. Author manuscript; available in PMC: 2017 Feb 15.
Published in final edited form as: Biochem J. 2016 Feb 15;473(4):347–364. doi: 10.1042/BJ20150942

Table 4.

Targeting ligands in PDT

Class Ligand Target PS Application Reference
Monoclonal antibody OC125 Ovarian cancer Chlorin(e6) Cancer, in vitro, in vivo [157]
Peptide Octreotide Somatostatin receptor Chlorin(e6) Leukaemia, in vitro [81]
Peptide RGD tripeptide αvβ3 integrin Phaeophorbide a Cancer, in vitro [76]
Lipoprotein Low-density lipoprotein LDL receptor Tetra-t-butyl silicon phthalocyanine Cancer, atherosclerosis, in vitro, in vivo [158]
Serum protein Transferrin Transferrin receptor Hematoporphyrin Cancer, in vitro [77]
Serum protein Modified albumin Scavenger receptor Chlorin(e6) Atherosclerosis, in vitro, in vivo [159]
Vitamin Folic acid Folate receptor Phaeophorbide a Cancer, in vitro [76]
Steroid Oestradiol Steroid receptor Phaeophorbide a Breast cancer, in vitro [160]
Carbohydrate Mannose Mannose receptor Meso-tetraphenylporphyrin Cancer, in vitro [161]