Table 2. Inhibitory activity of ABH derivatives.
| Inhibitor | IC50 (µM) | K i (µM) |
|---|---|---|
| ABH, S-isomer (L) | 1.3 ± 0.2 | 0.9 ± 0.1 |
| ABHPE, S-isomer (L) | 2.1 ± 0.3 | 1.4 ± 0.2 |
| ABHDP, racemic (DL) | 1.7 ± 0.4 | 1.1 ± 0.3 |
| Inhibitor | IC50 (µM) | K i (µM) |
|---|---|---|
| ABH, S-isomer (L) | 1.3 ± 0.2 | 0.9 ± 0.1 |
| ABHPE, S-isomer (L) | 2.1 ± 0.3 | 1.4 ± 0.2 |
| ABHDP, racemic (DL) | 1.7 ± 0.4 | 1.1 ± 0.3 |