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. 2016 Mar 16;72(Pt 4):300–306. doi: 10.1107/S2053230X16003630

Table 2. Inhibitory activity of ABH derivatives.

Inhibitor IC50M) K iM)
ABH, S-isomer (L) 1.3 ± 0.2 0.9 ± 0.1
ABHPE, S-isomer (L) 2.1 ± 0.3 1.4 ± 0.2
ABHDP, racemic (DL) 1.7 ± 0.4 1.1 ± 0.3