Table 7. Imidazopyrazines Merck Research Laboratories.
| ||
---|---|---|
Compd | R | IC50a (nM) |
58 | 650 | |
59 | 60 |
Expressed as the inhibition of MK2 ability to phosphorylate a peptide substrate.
| ||
---|---|---|
Compd | R | IC50a (nM) |
58 | 650 | |
59 | 60 |
Expressed as the inhibition of MK2 ability to phosphorylate a peptide substrate.