Table2.
Selected RAS-targeted clinical trials
| Drug | Target | Phase | Study population | Clinicaltrials.gov |
| Selumetinib | MEK | 3 | Second line stage 4 or stage 3B NSCLC | NCT01933932 |
| MEK162+erlotinib | MEK | 1 | Metastatic, failed prior therapies | NCT01859026 |
| Trametinib+momelotinib | MEK+JAK1/2 | 1 | Metastatic, progression after platinum based chemotherapy | NCT02258607 |
| PALBOCICLIB+PD-0325901 | CDK4/6+MEK | 1/2 | Metastatic, failed prior therapies | NCT02022982 |
| AZD2014+selumetinib | mTOR+MEK | 1/2 | Metastatic, failed prior therapies | NCT02583542 |