Table IV.
Optical agents targeting PSMA
Inhibitor | Entry | Linker | Fluorophore | Reference |
---|---|---|---|---|
![]() |
1 | No linker | IRDye78 | 98 |
2 | No linker | IRDye800CW | 99 | |
3 |
![]() |
IRDye800RS | 99 | |
4 |
![]() |
IRDye800CW | 99 | |
5 | ||||
6 | ||||
| ||||
![]() |
7 | No linker | 5-FAM-X | 40 |
8 | No linker | 5-FAM | 100 | |
9 | PEG3 | 5-FAM | 100 | |
| ||||
![]() |
10 | No linker | Cy5.5 | 101 |
| ||||
![]() |
11 |
![]() |
![]() |
73 |
12 |
![]() |
IRDye800CW | 102 | |
13 | IRDye800RS | 103 | ||
14 | ICG derivative | 103 | ||
15 | Cy7 | 103 | ||
16 | Cy5.5 | 103 | ||
17 | No linker | IRDye800CW | 103 | |
18 | IRDye800RS | 103 | ||
19 | ICG derivative | 103 | ||
20 | Cy7 | 103 | ||
21 | Cy5.5 | 103 | ||
22 | IRDye800CW | 103 | ||
23 |
![]() |
IRDye800RS | 103 | |
24 | ICG derivative | 103 | ||
25 | Cy7 | 103 | ||
26 | Cy5.5 | 103 | ||
27 |
![]() |
IRDye800CW | 107 | |
| ||||
![]() |
28 |
![]() |
FITC | 75 |
29 | Rhodamine B | 75 | ||
30 |
![]() |
DyLight 680 | 105 | |
31 | Alexa Fluor 647 | 105 | ||
32 | IRDye800CW | 105 | ||
33 | Amc-Ahx-Glu-Glu-Glu-Lys | IRDye800CW | 106 | |
| ||||
![]() |
34 |
![]() |
5(6)-FAM | 48 |