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. 2016 Feb 29;16:171–182. doi: 10.1007/s40256-016-0163-6

Table 2.

Direct oral anticoagulants in development for the prevention of stroke in atrial fibrillation worldwide

Drug Manufacturer Mechanism of action Phase of development Frequency of administration Clinical trial(s)
Dabigatran etexilate Boehringer Ingelheim Thrombin inhibitor Marketed Twice daily RE-LY
Apixaban Pfizer/Bristol-Myers Squibb Factor Xa inhibitor Marketed Twice daily ARISTOTLE, AVERROES
Rivaroxaban Bayer/Janssen Factor Xa inhibitor Marketed Once daily ROCKET-AF
Edoxaban Daiichi Sankyo Factor Xa inhibitor Marketed (not in Mexico) Once daily ENGAGE AF-TIMI 48