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. Author manuscript; available in PMC: 2016 May 12.
Published in final edited form as: J Med Chem. 2014 Aug 28;58(1):2–29. doi: 10.1021/jm401994c

Table 3.

In vitro and in vivo inhibition of DNL.

Compound no Rat EC50 (nM) In vivo DNL inhibition (%)
32 > 10000 Not determined
33 100 65
34 20 78
35 30 Not determined
36 42 73
37 609 34
38 27 73