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. 2016 Feb 24;7(5):465–469. doi: 10.1021/acsmedchemlett.5b00479

Table 3. SAR of the R5 Group.

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Potency measured in human embryonic kidney (HEK) cells in the presence of 10 μM DETA-NO.

a

The geometric mean of at least two repeated runs, unless stated otherwise.

b

Not determined due to incomplete concentration response. Maximal efficacy (%Emax) at 30 μM shown in parentheses.