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. Author manuscript; available in PMC: 2016 May 21.
Published in final edited form as: ACS Chem Biol. 2016 Mar 2;11(5):1313–1321. doi: 10.1021/acschembio.6b00167

Table 1.

Effects of LEDGF/p75 on BI/D EC50 Values for Inducing Aberrant IN Multimerization

[LEDGF] nM BI/D EC50, µMa
0 0.11 ± 0.0088
2 1.39 ± 0.18
10 2.62 ± 0.30
20 3.22 ± 0.33
50 4.29 ± 0.32
100 5.22 ± 0.27
200 7.02 ± 0.89
a

Average values from three idependent experiments are shown