(a).
| CYP2D6 | ||
|---|---|---|
| Substrates | Inhibitors | Inducers |
| Amphetamine | Amiodarone | Corticosteroids/ dexamethasone Delavirdine Protease inhibitors (indinavir, lopinavir/ritonavir, saquinavir) |
| Amitriptyline | Amitriptyline | |
| Aripiprazole | Bupropion | |
| Atomoxetine | Celecoxib | |
| Beta-blockers (selected) | Chlorpheniramine | |
| Carbamazepine | Chlorpromazine | |
| Carvedilol | Cinacalcet | |
| Chlorpheniramine | Chloroquine | |
| Chlorpromazine | Cimetidine | |
| Cinacalcet | Citalopram | |
| Clomipramine | Clomipramine | |
| Desipramine | Clemastine | |
| Dextromethorphan | Cocaine | |
| Doxazosin | Clozapine | |
| Flecainide | Desipramine | |
| Fluvoxamine | Diphenhydramine | |
| Haloperidol | Doxepin | |
| Hydrocodone | Doxorubicin | |
| Imipramine | Escitalopram | |
| Lidocaine | Duloxetine | |
| Metoclopramide | Fluoxetine | |
| Metoprolol | Fluphenazine | |
| Mexiletine | Fluvoxamine | |
| Nortriptyline | Haloperidol | |
| Ondansetron | Hydroxyzine | |
| Oxycodone | Lomustine | |
| Paroxetine | Methadone | |
| Perphenazine | Metoclopramide | |
| Primaquine | Mibefradil | |
| Promethazine | Nefazodone | |
| Risperidone | Norfloxacin | |
| Tamoxifen | Quinidine | |
| Thioridazine | Paroxetine | |
| Timolol | Perphenazine | |
| Tricyclic antidepressants | Propafenone | |
| Venlafaxine | Quinidine | |
| Yohimbine | Ranitidine | |
| Ritonavir | ||
| Sertraline | ||
| Sertindole | ||
| Terbinafine | ||
| Thioridazine | ||
| Ticlopidine | ||
| Tricyclic antidepressants | ||
| Venlafaxine | ||
| Vinblastine | ||
| Vinorelbine | ||