A) Relative fitness of CRISPRi essential gene knockdown strains (n = 289) with basal dcas9 expression (no xylose induction) grown on plates containing MAC-0170636, as determined by the ratio of normalized colony sizes on LB plates + DMSO versus LB + MAC-0170636.
B) Minimal inhibitory concentration (MIC) assay for strains over- or under-expressing uppS grown in liquid medium containing MAC-0170636. The MICs of these strains were (in μg/ml): sgRNAuppS + 0.05% xyl (∼0.012), sgRNAuppS (∼0.195), WT (∼0.78), and uppS overexpression (∼3.125). The values plotted are the means of at least three measurements, and error bars are ±1 standard deviation.
C) Concentration-dependent inhibition of purified B. subtilis UppS by MAC-0170636. Each point is an individual measurement.
D) MIC assay for strains expressing B. subtilis uppS (BsΔuppS/amyE∷Pspank-uppSBs) or S. aureus uppS (BsΔuppS/amyE∷Pspank-uppSSa) grown in liquid LB + MAC-0170636.