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. Author manuscript; available in PMC: 2016 Jun 7.
Published in final edited form as: Future Med Chem. 2016 Mar 15;8(4):463–489. doi: 10.4155/fmc.16.5

Table 2.

Published selective inhibitors of HSET and their biological activities

Compound Identifier Structure HSET Biochemical IC50 (nM)a References
CW069 17 graphic file with name emss-68393-i017.jpg 75000 [60]
AZ82 18 graphic file with name emss-68393-i018.jpg 310 [61]
a

IC50s determined in microtubule-stimulated biochemical assays.