Table 3. Some σR ligands in order of their potency.
σR ligands in rough order of potency | |
---|---|
σ1R ligands | σ2R ligands |
(+)-pentazocine [PTZ] | 1,3 di-o-tolyl-guanidine [DTG] |
Haloperidol | Haloperidol |
1,3 di-o-tolyl-guanidine [DTG] | (+)-3-PPP [preclamol) |
(+)-3-PPP | (−)-pentazocine |
Dextromethorphan [DEX] | Phencyclidine |
(+)-SKF 10,047 | (+)-pentazocine |
(+)-cyclazocine | (−)-SKF 10,047 |
(−)-pentazocine | BD1047 |
Phencyclidine | BD1063 |
(−)-SKF 10,047 |