Table 3. Some σR ligands in order of their potency.
| σR ligands in rough order of potency | |
|---|---|
| σ1R ligands | σ2R ligands |
| (+)-pentazocine [PTZ] | 1,3 di-o-tolyl-guanidine [DTG] |
| Haloperidol | Haloperidol |
| 1,3 di-o-tolyl-guanidine [DTG] | (+)-3-PPP [preclamol) |
| (+)-3-PPP | (−)-pentazocine |
| Dextromethorphan [DEX] | Phencyclidine |
| (+)-SKF 10,047 | (+)-pentazocine |
| (+)-cyclazocine | (−)-SKF 10,047 |
| (−)-pentazocine | BD1047 |
| Phencyclidine | BD1063 |
| (−)-SKF 10,047 | |