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. 2015 Jun 9;36(4):327–388. doi: 10.3109/10799893.2015.1015737

Table 3. Some σR ligands in order of their potency.

σR ligands in rough order of potency
σ1R ligands σ2R ligands
(+)-pentazocine [PTZ] 1,3 di-o-tolyl-guanidine [DTG]
Haloperidol Haloperidol
1,3 di-o-tolyl-guanidine [DTG] (+)-3-PPP [preclamol)
(+)-3-PPP (−)-pentazocine
Dextromethorphan [DEX] Phencyclidine
(+)-SKF 10,047 (+)-pentazocine
(+)-cyclazocine (−)-SKF 10,047
(−)-pentazocine BD1047
Phencyclidine BD1063
(−)-SKF 10,047